SCHEMBL28445488

SCHEMBL28445488

FC(F)(F)c1ccccc1CSc1nnc(CSc2nc3ccccc3s2)o1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.52
TSHR P16473 4/20 0.52
LMNA P02545 4/20 0.52
PIEZO1 Q92508 1/20 0.48
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 4/20 0.47
BACE1 P56817 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CASP1 P29466 1/20 0.47
RAB9A P51151 5/20 0.47
NPC1 O15118 3/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
MAPT P10636 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28446500 0.84 TSHR (0.58) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28445490 0.81 TSHR (0.57) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28453972 0.80 MAPK1 (0.54) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28452388 0.79 TSHR (0.49) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28449603 0.79 MAPK1 (0.49) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28448687 0.78 MGAM (0.54) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28448690 0.77 PTK2 (0.56) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28453905 0.76 ALDH1A1 (0.57) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28453935 0.75 PTK2 (0.56) MAPK1TSHRLMNAALDH1A1HSD17B10
SCHEMBL28452384 0.75 PTK2 (0.56) MAPK1TSHRLMNAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106916150-B 1,3, 4-oxadiazole-2-methylthio-benzothiazole derivative, preparation method and application thereof 中国科学院上海药物研究所 2020-08-25 CN claimed
CN-106916150-B 1,3, 4-oxadiazole-2-methylthio-benzothiazole derivative, preparation method and application thereof 中国科学院上海药物研究所 2020-08-25 CN disclosed