SCHEMBL28445812

SCHEMBL28445812

CC(C)(C)OC(=O)N[C@@H]1C[C@@H](C(F)(F)F)CC12CCNCC2

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.34
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
EPHX2 P34913 1/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18328497 1.00 BTK (0.34) BTKMEN1MAPK1KMT2AGAA
SCHEMBL21287726 0.87 BTK (0.37) BTKMEN1MAPK1KMT2AGAA
SCHEMBL21287164 0.84 BTK (0.37) BTKMEN1MAPK1KMT2AGAA
SCHEMBL23028470 0.84 CTSK (0.34) BTKMEN1MAPK1KMT2ANFKB1
SCHEMBL8319039 0.84 GAA (0.39) BTKMEN1MAPK1KMT2AGAA
SCHEMBL21287163 0.83 BTK (0.36) BTKMEN1MAPK1KMT2AGAA
SCHEMBL22814480 0.83 BTK (0.36) BTKMEN1MAPK1KMT2AGAA
SCHEMBL20337372 0.82 BTK (0.34) BTKMEN1MAPK1KMT2AEPHX2
SCHEMBL20337417 0.82 BTK (0.34) BTKMEN1MAPK1KMT2AEPHX2
SCHEMBL20337488 0.81 SSTR4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112625028-A Compounds and compositions for inhibiting SHP2 activity 诺华股份有限公司 2021-04-09 CN disclosed
CN-107922388-B Compounds and compositions for inhibiting SHP2 activity 诺华股份有限公司 2020-12-29 CN disclosed
CN-107787323-B Compounds and compositions for inhibiting SHP2 activity 诺华股份有限公司 2020-09-01 CN disclosed