SCHEMBL28446331

SCHEMBL28446331

CC(C)(C)OC(=O)NCCCCCCn1cc(-c2cccc(C(=O)O)n2)cn1.[LiH]

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 5/20 0.48
ACACB O00763 1/20 0.42
ACACA Q13085 1/20 0.42
DRD2 P14416 5/20 0.42
P2RY12 Q9H244 2/20 0.40
CYP3A4 P08684 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18012836 0.99 SUCNR1 (0.49) SUCNR1ACACBACACADRD2P2RY12
SCHEMBL17966554 0.91 SUCNR1 (0.46) SUCNR1ACACBACACADRD2P2RY12
Lithium Ion SCHEMBL17966543 0.90 SUCNR1 (0.46) SUCNR1ACACBACACADRD2P2RY12
SCHEMBL17966514 0.89 SUCNR1 (0.41) SUCNR1ACACBACACAP2RY12CKS1B
SCHEMBL18012770 0.88 SUCNR1 (0.42) SUCNR1ACACBACACAP2RY12CKS1B
SCHEMBL17998113 0.88 DRD2 (0.43) SUCNR1ACACBACACADRD2CYP3A4
SCHEMBL30875448 0.88 DRD2 (0.43) SUCNR1ACACBACACADRD2CYP3A4
Lithium SCHEMBL17966518 0.88 SUCNR1 (0.41) SUCNR1ACACBACACAP2RY12CKS1B
SCHEMBL17998112 0.83 CACNA1G (0.49) DRD2CYP3A4CKS1BSKP1SKP2
SCHEMBL19407199 0.83 DRD2 (0.42) SUCNR1ACACBACACADRD2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849055-B Macrocyclic compounds useful as IRAK1/4 inhibitors and uses thereof 默克专利有限公司 2020-08-07 CN disclosed