SCHEMBL28446552

SCHEMBL28446552

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55
ADRA1D P25100 1/20 0.55
ADRA1A P35348 1/20 0.55
ADRA1B P35368 1/20 0.55
TSHR P16473 2/20 0.54
PDE1C Q14123 2/20 0.54
ALDH1A1 P00352 3/20 0.53
HSD17B10 Q99714 2/20 0.53
KDM4E B2RXH2 2/20 0.53
HTT P42858 1/20 0.53
RAB9A P51151 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ADORA3 P0DMS8 1/20 0.52
CACNA1F O60840 2/20 0.52
CACNA1D Q01668 2/20 0.52
CACNA1S Q13698 2/20 0.52
CACNA1C Q13936 2/20 0.52
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035270 0.95 TSHR (0.59) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7386637 0.88 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7385666 0.88 ADRA2A (0.48) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL28435076 0.87 ADORA3 (0.67) ADRA1ATSHRALDH1A1HSD17B10KDM4E
SCHEMBL7379815 0.87 ADRA2A (0.45) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7380762 0.87 ADORA3 (0.51) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11784686 0.85 KMT2A (0.65) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7267420 0.83 CACNA1B (0.68) ADORA3CACNA1B
SCHEMBL7265410 0.82 TSHR (0.65) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL28440531 0.81 CACNA1B (0.44) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423362-A Preparation method of two high-purity clevidipine butyrate impurities 山东省药学科学院 2020-07-17 CN claimed
CN-111423362-A Preparation method of two high-purity clevidipine butyrate impurities 山东省药学科学院 2020-07-17 CN disclosed