SCHEMBL28447448

SCHEMBL28447448

O=C(OCCBr)c1ccc2c(c1)NCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.39
CRBN Q96SW2 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
JAK2 O60674 2/20 0.38
JAK3 P52333 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968115 0.83 JAK2 (0.51) ALDH1A1CYP2C9ALOX15CYP2C19JAK2
SCHEMBL3872066 0.83 JAK2 (0.51) ALDH1A1CYP2C9ALOX15CYP2C19JAK2
Hydrochloric Acid SCHEMBL27081766 0.82 JAK2 (0.50) ALDH1A1CYP2C9ALOX15CYP2C19JAK2
SCHEMBL12931800 0.80 SNCA (0.46) ACHECRBNALDH1A1CYP2C9ALOX15
Hydrochloric Acid SCHEMBL1271624 0.78 SNCA (0.45) ACHECRBNALDH1A1CYP2C9ALOX15
SCHEMBL30026444 0.78 KMT2A (0.53) ACHEALDH1A1SMN1; SMN2MAPTKDM4E
SCHEMBL29906783 0.78 ALDH1A1 (0.47) CRBNALDH1A1ALOX15HDAC3HDAC4
SCHEMBL2898350 0.78 ALDH1A1 (0.47) CRBNALDH1A1ALOX15HDAC3HDAC4
Hydrochloric Acid SCHEMBL29940234 0.77 ALDH1A1 (0.46) CRBNALDH1A1ALOX15HDAC3HDAC4
Hydrochloric Acid SCHEMBL3102567 0.77 ALDH1A1 (0.46) CRBNALDH1A1ALOX15HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074816-B Heterocyclic derivative, preparation method and medical application thereof 四川海思科制药有限公司 2020-07-17 CN disclosed