SCHEMBL28447680

SCHEMBL28447680

C=CC(=O)Nc1cccc(Nc2nc(Cl)ncc2-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.55
EGFR P00533 11/20 0.54
JAK2 O60674 3/20 0.54
JAK3 P52333 3/20 0.54
ITK Q08881 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9924738 0.88 BTK (0.69) BTKEGFRJAK2JAK3
SCHEMBL28447678 0.85 BTK (0.53) BTKEGFRJAK2JAK3ITK
SCHEMBL15814594 0.80 EGFR (0.74) BTKEGFRJAK2JAK3ITK
SCHEMBL9945478 0.80 BTK (0.67) BTKEGFR
SCHEMBL28445845 0.79 EGFR (0.60) BTKEGFRITK
SCHEMBL9923766 0.78 BTK (0.74) BTKEGFRITK
SCHEMBL9945480 0.78 BTK (0.69) BTKEGFRITK
SCHEMBL18970176 0.77 BTK (0.60) BTKEGFRJAK2JAK3ITK
SCHEMBL28059334 0.77 BTK (0.85) BTKEGFRJAK2JAK3ITK
SCHEMBL12519708 0.77 BTK (0.82) BTKEGFRJAK2JAK3ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed