SCHEMBL28445845

SCHEMBL28445845

C=CC(=O)Nc1cccc(Nc2nc(Cl)ncc2OC(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.60
ITK Q08881 7/20 0.60
BTK Q06187 5/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16370843 0.86 EGFR (0.73) EGFRITKBTK
SCHEMBL9924738 0.84 BTK (0.69) EGFRBTK
SCHEMBL28455992 0.84 EGFR (0.66) EGFRITKBTK
SCHEMBL28446232 0.83 SYK (0.54) EGFRITK
SCHEMBL15814594 0.83 EGFR (0.74) EGFRITKBTK
SCHEMBL9945478 0.82 BTK (0.67) EGFRBTK
SCHEMBL9923766 0.81 BTK (0.74) EGFRITKBTK
SCHEMBL9945480 0.81 BTK (0.69) EGFRITKBTK
SCHEMBL28447678 0.79 BTK (0.53) EGFRITKBTK
SCHEMBL28447680 0.79 BTK (0.55) EGFRITKBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed