SCHEMBL28451635

SCHEMBL28451635

CNc1cc(-c2ncc(C(F)(F)F)cn2)ncn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.52
CYP3A4 P08684 1/20 0.52
CLK4 Q9HAZ1 2/20 0.43
CYP2D6 P10635 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
ABL1 P00519 2/20 0.40
BCR P11274 2/20 0.40
JAK2 O60674 2/20 0.40
EGFR P00533 1/20 0.40
JAK1 P23458 1/20 0.39
TNNI3K Q59H18 4/20 0.36
KDR P35968 3/20 0.36
MAPK14 Q16539 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28447698 0.98 CYP1A2 (0.51) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL16894166 0.77 ABL1 (0.61) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL16894261 0.76 ABL1 (0.59) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28074525 0.74 CYP1A2 (0.52) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28242142 0.73 CYP1A2 (0.58) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28451607 0.72 MAPK1 (0.37) KMT2ATNNI3KKDRMAPK14BRAF
SCHEMBL17979199 0.71 NPC1 (0.33) ALDH1A1KMT2A
SCHEMBL28451814 0.71 CYP1A2 (0.49) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28017373 0.71 ABL1 (0.55) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL18047668 0.70 NPC1 (0.32) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476640-B Bicyclic proline compounds 豪夫迈·罗氏有限公司 2022-02-25 CN disclosed
CN-107922392-B 1- (hetero) arylsulfonyl- (pyrrolidine or piperidine) -2-carboxamide derivatives and uses thereof 豪夫迈·罗氏有限公司 2020-07-21 CN disclosed