SCHEMBL28074525

SCHEMBL28074525

CNc1cc(-c2cnc(C(F)(F)F)nc2)ncn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.52
CYP3A4 P08684 1/20 0.52
CLK4 Q9HAZ1 2/20 0.43
CYP2D6 P10635 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
ABL1 P00519 5/20 0.40
BCR P11274 5/20 0.40
JAK2 O60674 3/20 0.40
KDR P35968 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
EGFR P00533 1/20 0.34
FAAH O00519 1/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664909 0.81 CYP1A2 (0.43) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28017373 0.80 ABL1 (0.55) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL22838564 0.80 CYP1A2 (0.51) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL28017385 0.79 ABL1 (0.54) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL16894166 0.77 ABL1 (0.61) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL21442182 0.77 TRPA1 (0.46) TRPV3
Hydrochloric Acid SCHEMBL16894261 0.76 ABL1 (0.59) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL16635390 0.75 AAK1 (0.39) CLK4ALDH1A1ABL1BCRTRPV3
SCHEMBL22838720 0.74 CYP1A2 (0.46) CYP1A2CYP3A4CLK4CYP2D6HSD17B10
SCHEMBL28451635 0.74 CYP1A2 (0.52) CYP1A2CYP3A4CLK4CYP2D6HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed