SCHEMBL28451607

SCHEMBL28451607

CNC(=O)Oc1cc(-c2ncc(C(F)(F)F)cn2)ncn1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.37
POLB P06746 2/20 0.36
PKM P14618 2/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 1/20 0.36
SCN9A Q15858 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
KDR P35968 4/20 0.33
MAPK14 Q16539 4/20 0.33
TNNI3K Q59H18 4/20 0.33
BRAF P15056 2/20 0.33
GAA P10253 1/20 0.33
AGBL2 Q5U5Z8 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28451635 0.72 CYP1A2 (0.52) KMT2ATRPV1KDRMAPK14TNNI3K
SCHEMBL1936666 0.71 ALDH1A1 (0.39) MAPK1PKMKMT2ALMNAKDR
Hydrochloric Acid SCHEMBL28447698 0.71 CYP1A2 (0.51) KMT2ATRPV1KDRMAPK14TNNI3K
SCHEMBL18018332 0.70 CACNA1H (0.43) POLBGAA
SCHEMBL18047666 0.69 KCNH2 (0.38) MAPK1POLBKMT2ALMNAGAA
SCHEMBL22582959 0.68 MAPK1 (0.43) MAPK1POLBPKMKMT2AGAA
SCHEMBL22583410 0.68 MAPK1 (0.49) MAPK1POLBPKMKMT2ALMNA
SCHEMBL18047664 0.68 TRPA1 (0.40) AGBL2
SCHEMBL16161634 0.67 KMO (0.54) PKMLMNAMAPT
SCHEMBL28442827 0.63 MAPT (0.34) POLBPKMKDRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476640-B Bicyclic proline compounds 豪夫迈·罗氏有限公司 2022-02-25 CN disclosed
CN-107922392-B 1- (hetero) arylsulfonyl- (pyrrolidine or piperidine) -2-carboxamide derivatives and uses thereof 豪夫迈·罗氏有限公司 2020-07-21 CN disclosed