SCHEMBL28451986

SCHEMBL28451986

O=C(CNc1cc(Br)cc2[nH]ncc12)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 19/20 0.55
IDO1 P14902 18/20 0.55
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19249344 0.88 TDO2 (0.51) TDO2IDO1CYP2C9
SCHEMBL28447373 0.86 IDO1 (0.50) TDO2IDO1CYP2C9
SCHEMBL19249343 0.82 TDO2 (0.74) TDO2IDO1CYP2C9
SCHEMBL19248997 0.80 NPC1 (0.52) TDO2IDO1
SCHEMBL28457353 0.80 TDO2 (0.59) TDO2IDO1CYP2C9
SCHEMBL28451310 0.78 TDO2 (0.64) TDO2IDO1CYP2C9
SCHEMBL19248990 0.75 TDO2 (0.72) TDO2IDO1
SCHEMBL22083965 0.75 TDO2 (0.69) TDO2IDO1CYP2C9
SCHEMBL28451309 0.71 TDO2 (0.52) TDO2IDO1CYP2C9
SCHEMBL19249342 0.71 TDO2 (0.52) TDO2IDO1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107033087-B 1H-indazole-4-amine compounds and use thereof as IDO inhibitors 西华大学 2020-09-04 CN disclosed