SCHEMBL28453047

SCHEMBL28453047

O=Cc1nc2c(s1)CCN(C(=O)O)C2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.33
DPP8 Q6V1X1 4/20 0.33
DPP7 Q9UHL4 4/20 0.33
DPP9 Q86TI2 3/20 0.33
GRM5 P41594 6/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779792 0.88 GRM5 (0.42) GRM5NPC1RAB9AMAPK1
SCHEMBL25390011 0.80 GRM5 (0.34) DPP4DPP8DPP7DPP9GRM5
SCHEMBL28449516 0.78 DRD2 (0.43) DPP4DPP8DPP7DPP9GRM5
SCHEMBL5642534 0.75 DPP4 (0.50) DPP4DPP8DPP7DPP9GRM5
SCHEMBL26094092 0.69 ADORA1 (0.40)
SCHEMBL3441635 0.68 HDAC6 (0.43)
SCHEMBL15332856 0.68 PDK1 (0.48) GRM5NPC1RAB9A
SCHEMBL15896560 0.68 PDK1 (0.48) GRM5NPC1RAB9A
SCHEMBL17377204 0.68 CSNK2A2 (0.41) NPC1RAB9AMAPK1
SCHEMBL21040978 0.67 ADORA1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922430-B 2-substituted benzimidazole-4-formamide compound and preparation method and application thereof 中国科学院上海药物研究所 2020-09-04 CN disclosed