SCHEMBL28454459

SCHEMBL28454459

c1csc(-c2n[nH]nc2-c2cccs2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB2 Q9UBS0 5/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.47
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44
CASP1 P29466 1/20 0.44
RAB9A P51151 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NISCH Q9Y2I1 1/20 0.44
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2373414 0.78 MEN1 (0.42) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL2218274 0.75 RPS6KB2 (0.50) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL820251 0.75 RPS6KB2 (0.50) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL16291133 0.74 L3MBTL1 (0.57) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL3545 0.74 L3MBTL1 (0.57) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL2877926 0.73 ADORA2A (0.42) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL2049905 0.73 RPS6KB2 (0.41) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL3473292 0.73 RPS6KB2 (0.41) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL11624487 0.73 RPS6KB2 (0.44) RPS6KB2MEN1KMT2AKDM4EALDH1A1
SCHEMBL623377 0.72 MAPT (0.41) RPS6KB2MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438376-B 4, 5-diheteroaryl substituted triazole compound and preparation method and application thereof 扬州工业职业技术学院 2020-09-04 CN disclosed