SCHEMBL28459484

SCHEMBL28459484

CC(C)(O)C(O)Nc1nc(Cl)nc(Nc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.65
IDH2 P48735 11/20 0.60
LMNA P02545 2/20 0.51
MAPT P10636 2/20 0.51
MAPK1 P28482 1/20 0.51
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28455014 0.82 IDH2 (0.88) APPIDH2LMNAMAPTMAPK1
SCHEMBL30568814 0.82 APP (0.79) APPIDH2LMNAMAPTMAPK1
SCHEMBL1391344 0.82 APP (0.79) APPIDH2LMNAMAPTMAPK1
SCHEMBL28455336 0.81 IDH2 (0.88) APPIDH2
SCHEMBL28458402 0.81 IDH2 (0.85) APPIDH2LMNAMAPTMAPK1
SCHEMBL13771505 0.79 APP (0.76) APPIDH2LMNAMAPTMAPK1
SCHEMBL28451054 0.77 IDH2 (0.89) APPIDH2LMNAMAPTMAPK1
SCHEMBL28456839 0.77 IDH2 (0.89) APPIDH2LMNAMAPTMAPK1
SCHEMBL28460991 0.77 IDH2 (0.89) APPIDH2LMNAMAPTMAPK1
SCHEMBL28447648 0.75 IDH2 (1.00) APPIDH2LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed