SCHEMBL28457809

SCHEMBL28457809

COc1ccc2c(c1)CCc1c(-c3cnccn3)c[nH]c1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.44
CYP17A1 P05093 1/20 0.44
CYP11B2 P19099 8/20 0.44
CYP11B1 P15538 4/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
MIF P14174 2/20 0.42
MEN1 O00255 1/20 0.41
ALPL P05186 1/20 0.41
CLK1 P49759 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 1/20 0.39
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5814304 0.79 EGFR (0.52) CYP19A1CYP17A1CYP11B2CYP1A2CYP2D6
SCHEMBL29899282 0.79 EGFR (0.52) CYP19A1CYP17A1CYP11B2CYP1A2CYP2D6
SCHEMBL28460940 0.79 CYP19A1 (0.41) CYP19A1CYP17A1CYP11B2CYP11B1
SCHEMBL5809047 0.77 ACHE (0.46) CYP19A1CYP11B2CYP1A2CYP2D6KDM4E
SCHEMBL30149529 0.77 ACHE (0.46) CYP19A1CYP11B2CYP1A2CYP2D6KDM4E
SCHEMBL28456202 0.76 CYP1A2 (0.49) CYP19A1CYP17A1CYP11B2CYP1A2CYP2D6
SCHEMBL28461711 0.73 EGFR (0.44) CYP19A1CYP17A1CYP11B2CYP1A2CYP2D6
SCHEMBL28454236 0.72 CYP1A2 (0.46) CYP19A1CYP17A1CYP11B2CYP11B1CYP1A2
SCHEMBL5419686 0.71 MAPK1 (0.49) CYP19A1CYP11B2CYP11B1CYP2D6KDM4E
SCHEMBL31140253 0.71 CYP1A1 (0.51) CYP11B2CYP11B1CYP1A2CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110283159-B 2, 4-disubstituted pyrrole or 2,3, 4-trisubstituted pyrrole prepared by one-pot method and preparation method thereof 河南大学 2020-09-29 CN disclosed