SCHEMBL28460940

SCHEMBL28460940

c1ccc2c(c1)CCc1c(-c3cnccn3)c[nH]c1-2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.41
CYP11B2 P19099 10/20 0.41
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
CDC42BPB Q9Y5S2 1/20 0.39
ADRA1D P25100 1/20 0.39
CYP11B1 P15538 7/20 0.39
LRRK2 Q5S007 1/20 0.38
NPC1 O15118 1/20 0.37
CYP17A1 P05093 1/20 0.36
DYRK1A Q13627 1/20 0.35
METAP2 P50579 1/20 0.35
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
HASPIN Q8TF76 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28457809 0.79 CYP19A1 (0.44) CYP19A1CYP11B2CYP11B1CYP17A1
SCHEMBL4155429 0.70 CYP19A1 (0.48) CYP19A1CYP11B2ADRA1AADRA1BADRA1D
SCHEMBL23649351 0.69 NPC1 (0.40) CYP19A1CYP11B2CYP11B1NPC1CYP17A1
SCHEMBL12853973 0.69 ALOX5AP (0.50) CYP19A1CYP11B2ADRA1AADRA1BADRA1D
SCHEMBL12853984 0.69 ALOX5AP (0.50) CYP19A1CYP11B2ADRA1AADRA1BADRA1D
SCHEMBL7705613 0.68 NOS3 (0.45) CYP19A1CYP11B2ADRA1AADRA1BADRA1D
SCHEMBL28462071 0.68 PARP1 (0.40) CYP11B2CYP11B1NPC1
SCHEMBL23064176 0.67 HSD17B10 (0.56) NPC1DYRK1AMETAP2
SCHEMBL28462072 0.67 NPC1 (0.36) CYP19A1CYP11B2CYP11B1NPC1DYRK1A
SCHEMBL4073407 0.67 ADRA1A (0.43) ADRA1AADRA1BROCK2ROCK1CDC42BPB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110283159-B 2, 4-disubstituted pyrrole or 2,3, 4-trisubstituted pyrrole prepared by one-pot method and preparation method thereof 河南大学 2020-09-29 CN disclosed