SCHEMBL28458039

SCHEMBL28458039

CCOC(=O)c1nc2c([N+](=O)[O-])cccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.47
PKN2 Q16513 1/20 0.47
GAA P10253 2/20 0.45
MGAM O43451 1/20 0.45
SI P14410 1/20 0.45
MGAM2 Q2M2H8 1/20 0.45
CACNA1C Q13936 2/20 0.44
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
MAPT P10636 2/20 0.43
NFKB1 P19838 1/20 0.43
MAPK1 P28482 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
PARP1 P09874 1/20 0.42
CYP1A2 P05177 1/20 0.42
CHEK1 O14757 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8277810 0.81 PKN1 (0.53) PKN1PKN2GAAMGAMSI
SCHEMBL8601951 0.80 PKN1 (0.55) PKN1PKN2GAAMGAMSI
SCHEMBL8598655 0.79 PKN1 (0.53) PKN1PKN2GAAMGAMSI
SCHEMBL7480899 0.78 PKN1 (0.50) PKN1PKN2GAAMGAMSI
SCHEMBL1013588 0.76 PKN1 (0.60) PKN1PKN2GAAMGAMSI
SCHEMBL7259082 0.76 GAA (0.65) PKN1PKN2GAAMGAMSI
Dimethylamine SCHEMBL7486960 0.76 PKN1 (0.56) PKN1PKN2GAAMGAMSI
SCHEMBL9588046 0.75 PARP1 (0.42) GAARAB9ANPC1MAPTALDH1A1
SCHEMBL28467668 0.74 PKN1 (0.49) PKN1PKN2GAAMGAMSI
SCHEMBL8598342 0.74 GAA (0.56) PKN1PKN2GAAMGAMSI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098846-B N-acyl sulfonamide FBPase inhibitor, preparation method thereof, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-10-09 CN disclosed