SCHEMBL7259082

SCHEMBL7259082

CCOC(=O)c1cccc2[nH]c(-c3ccccc3[N+](=O)[O-])nc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.65
MGAM O43451 1/20 0.65
SI P14410 1/20 0.65
MGAM2 Q2M2H8 1/20 0.65
PARP1 P09874 7/20 0.52
PRKD3 O94806 1/20 0.48
MAP4K4 O95819 1/20 0.48
PIM1 P11309 1/20 0.48
CLK2 P49760 1/20 0.48
MAP4K2 Q12851 1/20 0.48
CAMK2D Q13557 1/20 0.48
DYRK1A Q13627 1/20 0.48
PIM3 Q86V86 1/20 0.48
AURKB Q96GD4 1/20 0.48
PRKD2 Q9BZL6 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
STK17A Q9UEE5 1/20 0.48
MAP4K5 Q9Y4K4 1/20 0.48
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29412040 0.82 PARP1 (0.66) GAAMGAMSIMGAM2PARP1
SCHEMBL3580402 0.82 PARP1 (0.69) GAAPARP1PRKD3MAP4K4PIM1
SCHEMBL3574922 0.80 PARP1 (0.56) PARP1PRKD3MAP4K4PIM1CLK2
SCHEMBL6948231 0.79 PARP1 (0.69) PARP1PRKD3MAP4K4PIM1CLK2
SCHEMBL6511414 0.79 MGAM (1.00) GAAMGAMSIMGAM2PKN1
SCHEMBL6170661 0.78 PARP1 (0.64) PARP1PRKD3MAP4K4PIM1CLK2
SCHEMBL7718410 0.77 MGAM (0.69) GAAMGAMSIMGAM2PARP1
SCHEMBL7259179 0.77 ALDH1A1 (0.47) GAAPARP1ALDH1A1MAPTSMN1; SMN2
SCHEMBL28458039 0.76 PKN1 (0.47) GAAMGAMSIMGAM2PARP1
SCHEMBL9044494 0.76 MGAM (0.71) GAAMGAMSIMGAM2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057667-A2 STRAPPED AND MODIFIED BIS (BENZIMIDAZOLE) DIAMIDES FOR ASYMMETRIC CATALYSTS AND OTHER APPLICATIONS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2003-07-17 WO disclosed