SCHEMBL28458193

SCHEMBL28458193

COc1ccc2nc(-c3ccccc3)c(OCc3ccc(Br)cc3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.53
MAOB P27338 1/20 0.49
ALDH1A1 P00352 4/20 0.46
LMNA P02545 4/20 0.46
KDM4E B2RXH2 4/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
MAPT P10636 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
POLB P06746 1/20 0.46
NQO2 P16083 1/20 0.46
RAB9A P51151 1/20 0.46
PRNP P04156 1/20 0.45
HTT P42858 1/20 0.45
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28458555 0.87 ALDH1A1 (0.44) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL28450170 0.79 ALDH1A1 (0.50) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL14144076 0.77 MAPK14 (0.62) GPBAR1ALDH1A1LMNAKDM4EL3MBTL1
SCHEMBL31070199 0.77 KDM4E (0.74) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL8112450 0.77 KDM4E (0.74) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL6304505 0.71 KDM4E (0.62) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL28459393 0.71 ALDH1A1 (0.60) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL932888 0.70 PRNP (0.49) ALDH1A1LMNAKDM4EL3MBTL1NPSR1
SCHEMBL28430136 0.70 CFTR (0.57) GPBAR1ALDH1A1LMNAMEN1KMT2A
SCHEMBL29388744 0.70 CFTR (0.57) GPBAR1ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499585-B Quinoxaline derivative and preparation method and application thereof 浙江工业大学 2022-02-22 CN disclosed
CN-111499585-A Quinoxaline derivative and preparation method and application thereof 浙江工业大学 2020-08-07 CN disclosed