SCHEMBL28458399

SCHEMBL28458399

O=C(O)c1cccc2onc(C(=O)O)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 3/20 0.43
TSHR P16473 3/20 0.43
ALOX15 P16050 2/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
AGER Q15109 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
AURKB Q96GD4 5/20 0.42
PTPN1 P18031 1/20 0.41
HIF1A Q16665 2/20 0.41
CYP1A2 P05177 1/20 0.40
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
USP2 O75604 1/20 0.37
DUSP3 P51452 1/20 0.36
NR4A1 P22736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31754870 0.81 DUSP3 (0.41) ALDH1A1KDM4EHSD17B10AURKBPTPN1
SCHEMBL6830612 0.78 KCNA5 (0.48) KDM4EMAPTL3MBTL1PTPN1HIF1A
SCHEMBL496601 0.72 HIF1A (0.65) PTPN1HIF1A
SCHEMBL70977 0.69 HSD17B10 (0.48) ALDH1A1KDM4ETSHRALOX15HSD17B10
SCHEMBL13701003 0.68 AURKB (0.46) ALDH1A1KDM4EMAPTL3MBTL1AURKB
SCHEMBL4243185 0.68 KDM4E (0.47) ALDH1A1KDM4ETSHRALOX15CYP3A4
SCHEMBL29685650 0.67 ALDH1A1 (0.54) ALDH1A1KDM4ETSHRALOX15HSD17B10
SCHEMBL516363 0.67 ALDH1A1 (0.54) ALDH1A1KDM4ETSHRALOX15HSD17B10
SCHEMBL4243184 0.66 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRALOX15HSD17B10
SCHEMBL29404347 0.65 HSD17B10 (0.78) ALDH1A1KDM4ETSHRALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111233852-A NON type chiral bisoxazoline ligand and synthetic method and application thereof 上海师范大学 2020-06-05 CN disclosed