SCHEMBL28458402

SCHEMBL28458402

FC(F)(F)c1cccc(Nc2nc(Cl)nc(Nc3ccccc3)n2)c1

nearest known ligand 0.85

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 6/20 0.85
APP P05067 4/20 0.82
MAPT P10636 3/20 0.65
MAPK1 P28482 2/20 0.65
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
CTSC P53634 1/20 0.64
AURKA O14965 1/20 0.61
LMNA P02545 3/20 0.60
NFKB1 P19838 1/20 0.60
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1391344 0.92 APP (0.79) IDH2APPMAPTMAPK1CTSC
SCHEMBL30568814 0.92 APP (0.79) IDH2APPMAPTMAPK1CTSC
SCHEMBL28455381 0.87 IDH2 (0.91) IDH2APPMAPTMAPK1MEN1
SCHEMBL13771505 0.86 APP (0.76) IDH2APPMAPTMAPK1CTSC
SCHEMBL30933618 0.86 APP (0.66) IDH2APPMAPTMAPK1CTSC
SCHEMBL30933619 0.86 APP (0.66) IDH2APPMAPTMAPK1CTSC
SCHEMBL30568792 0.84 APP (0.67) IDH2APPMAPTMAPK1CTSC
SCHEMBL28897970 0.84 APP (0.67) IDH2APPMAPTMAPK1CTSC
SCHEMBL2856487 0.83 IDH2 (0.71) IDH2APPMAPTMAPK1CTSC
SCHEMBL28455014 0.82 IDH2 (0.88) IDH2APPMAPTMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed