SCHEMBL28459557

SCHEMBL28459557

[c]1cc(-n2ccnc2)c[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
ENPP2 Q13822 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
NOTUM Q6P988 1/20 0.44
CYP2A6 P11509 1/20 0.43
BAZ2B Q9UIF8 1/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP19A1 P11511 2/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
IDO1 P14902 1/20 0.40
CYP51A1 Q16850 1/20 0.38
ADH5 P11766 2/20 0.37
PDE3B Q13370 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3695247 0.73 VHL (0.31) MAPT
SCHEMBL16673120 0.69 CYP3A4 (0.62) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL2532397 0.69 LMNA (0.78) CYP3A4LMNAMAPTENPP2MKNK1
Hydrochloric Acid SCHEMBL28701756 0.68 LMNA (0.75) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL22402234 0.67 CYP3A4 (0.53) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL3250899 0.66 CYP3A4 (0.71) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL161573 0.65 CYP3A4 (0.63) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL242819 0.65 CYP3A4 (0.47) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL18228239 0.65 CYP3A4 (0.52) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL3527180 0.65 CYP3A4 (0.38) CYP3A4LMNAMAPTENPP2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107629059-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-07-28 CN disclosed