SCHEMBL28459583

SCHEMBL28459583

CC(C)c1ccc2c(c1)CCCN2C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.64
PDK2 Q15119 1/20 0.64
PDK3 Q15120 1/20 0.64
PDK4 Q16654 1/20 0.64
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.47
NPSR1 Q6W5P4 3/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TP53 P04637 3/20 0.45
LMNA P02545 2/20 0.45
IDO1 P14902 2/20 0.45
KCNH2 Q12809 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 5/20 0.44
TSHR P16473 2/20 0.44
GRM7 Q14831 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13711475 0.88 PDK1 (0.64) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL17368396 0.87 PDK1 (0.62) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL6124252 0.86 PDK1 (0.61) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL22397647 0.84 KDM4E (0.51) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL24511819 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL22482270 0.81 PDK1 (0.57) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL4026091 0.80 KDM4E (0.71) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL28700900 0.79 NOTUM (0.49) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL28936707 0.79 NOTUM (0.49) PDK1PDK2PDK3PDK4HTR2A
SCHEMBL6626359 0.79 NOTUM (0.49) PDK1PDK2PDK3PDK4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111670034-A Pyranopyrazoles and pyrazolopyridines immunomodulators for the treatment of autoimmune diseases 洛克菲勒大学 2020-09-15 CN disclosed