SCHEMBL28459657

SCHEMBL28459657

O=C(NCc1ccccc1)c1c([N+](=O)[O-])c(NCc2ccccc2)nc2ccc(F)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.47
MAPT P10636 4/20 0.47
KMT2A Q03164 4/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
CYP1A2 P05177 1/20 0.45
PPARG P37231 1/20 0.44
LMNA P02545 2/20 0.43
MAPK1 P28482 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 3/20 0.43
POLB P06746 3/20 0.43
ALDH1A1 P00352 3/20 0.43
PDE5A O76074 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
RECQL P46063 1/20 0.43
RAB9A P51151 1/20 0.43
MCL1 Q07820 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28462514 0.95 HTT (0.47) EGFRMAPTKMT2AL3MBTL1LMNA
SCHEMBL28462518 0.93 EGFR (0.46) EGFRMAPTKMT2AL3MBTL1CYP1A2
SCHEMBL28471314 0.90 MEN1 (0.54) EGFRMAPTKMT2AL3MBTL1LMNA
SCHEMBL28466749 0.89 PTGER4 (0.45) EGFRALDH1A1HTTCTNNB1TCF7L2
SCHEMBL28465230 0.89 S1PR3 (0.42) EGFRMAPTKMT2AL3MBTL1LMNA
SCHEMBL28465234 0.89 EGFR (0.59) EGFRMAPTKMT2AL3MBTL1LMNA
SCHEMBL28460390 0.88 EGFR (0.55) EGFRMAPTKMT2AL3MBTL1PPARG
SCHEMBL28463573 0.88 LMNA (0.48) EGFRMAPTKMT2APPARGLMNA
SCHEMBL28462520 0.87 CTNNB1 (0.58) EGFRKMT2AL3MBTL1CYP1A2LMNA
SCHEMBL28470826 0.86 ALDH1A1 (0.54) MAPTKMT2AL3MBTL1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107522659-B 3-nitroquinoline derivative and preparation method and application thereof 云南大学 2020-09-29 CN disclosed