SCHEMBL28463524

SCHEMBL28463524

O=S1(=O)CCNCc2cc(Cl)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.50
HTR2C P28335 6/20 0.41
HTR2A P28223 5/20 0.41
HTR2B P41595 3/20 0.41
CHEK1 O14757 1/20 0.37
DAPK3 O43293 1/20 0.37
MAP4K4 O95819 1/20 0.37
RET P07949 1/20 0.37
PIM1 P11309 1/20 0.37
LTK P29376 1/20 0.37
GRK5 P34947 1/20 0.37
CSNK1A1 P48729 1/20 0.37
CDK8 P49336 1/20 0.37
PRKX P51817 1/20 0.37
LIMK1 P53667 1/20 0.37
CDK5 Q00535 1/20 0.37
ACVR1 Q04771 1/20 0.37
PTK2 Q05397 1/20 0.37
TYRO3 Q06418 1/20 0.37
PRKAA1 Q13131 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28438076 0.87 PNMT (0.50) PNMTHTR2CHTR2AHTR2BCHEK1
SCHEMBL2589655 0.75 CD44 (0.45) PNMTHTR2C
Hydrochloric Acid SCHEMBL5849050 0.74 CD44 (0.44) PNMTHTR2C
SCHEMBL31332057 0.70 CHRNB2 (0.41) HTR2CHTR2A
SCHEMBL329775 0.67 PNMT (1.00) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL532012 0.67 PNMT (0.85) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL29587836 0.67 PNMT (1.00) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL28445860 0.67 PNMT (0.49) PNMTHTR2CHTR2ARETGRK5
SCHEMBL31332153 0.67 CHRNB2 (0.41) HTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL1124954 0.66 PNMT (0.96) PNMTHTR2CHTR2AHTR2BASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111548325-A Preparation method of halogenated benzothiazepine compound, product prepared by preparation method and application of product 西安都创医药科技有限公司 2020-08-18 CN disclosed
CN-111548325-A Preparation method of halogenated benzothiazepine compound, product prepared by preparation method and application of product 西安都创医药科技有限公司 2020-08-18 CN disclosed