SCHEMBL28465962

SCHEMBL28465962

CCCC=C(CC)NC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.38
CA7 P43166 2/20 0.38
CA12 O43570 1/20 0.38
CA14 Q9ULX7 1/20 0.38
TDP1 Q9NUW8 1/20 0.34
CTSK P43235 14/20 0.34
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CTSS P25774 1/20 0.33
CA2 P00918 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19978200 0.86 CA1 (0.37) CA1CA7CA12CA14TDP1
SCHEMBL24223538 0.82 CTSK (0.40) CA1CA7CA12CA14TDP1
SCHEMBL19978301 0.80 CA1 (0.38) CA1CA7CA12CA14CTSK
SCHEMBL10011981 0.78 CA12 (0.37) CA1CA7CA12CA14CTSK
SCHEMBL19823872 0.77 CA1 (0.36) CA1CA7CA12CA14TDP1
Butanal SCHEMBL5051895 0.77 ALDH1A1 (0.46) CA1CA7CA12CA14TDP1
SCHEMBL19978199 0.76 CA1 (0.35) CA1CA7CA12CA14TDP1
SCHEMBL22168208 0.73 CA1 (0.35) CA1CA7CA12CA14TDP1
SCHEMBL28464582 0.71 EPHX1 (0.38) KMT2AALDH1A1CA2MEN1
SCHEMBL240769 0.71 CA1 (0.42) CA1CA7CA12CA14TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106795147-B Cyclopropyl fused thiazine-2-amine compounds as beta-secretase inhibitors and methods of use 美国安进公司 2020-09-22 CN disclosed