SCHEMBL28469141

SCHEMBL28469141

CC(C)(C)OC(=O)N1C[C@H](O)CC1(c1cc(F)ccc1F)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 3/20 0.37
APP P05067 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
DRD2 P14416 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
SLC6A2 P23975 1/20 0.37
HRH2 P25021 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR7 P34969 1/20 0.37
DRD3 P35462 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
SLC6A3 Q01959 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17830897 0.77 PSEN1 (0.38) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL1429735 0.74 PSEN1 (0.42) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL17353253 0.73 PSEN1 (0.42) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL21136075 0.72 RORC (0.42) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL20119114 0.72 PSEN1 (0.36) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL23327641 0.71 HSD11B1 (0.43) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL29891503 0.71 PSEN1 (0.41) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL21136665 0.71 PSEN1 (0.41) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL26465788 0.71 PSEN1 (0.41) PSEN1APPHTR1AADRA2ADRD2
SCHEMBL17848942 0.70 PSEN1 (0.33) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109890820-B Aminopyrazolopyrimidine compounds as neurotrophin tyrosine kinase receptor inhibitors 正大天晴药业集团股份有限公司 2020-11-03 CN disclosed
CN-108003161-B Neurotrophic factor tyrosine kinase receptor inhibitors 正大天晴药业集团股份有限公司 2020-10-09 CN disclosed