SCHEMBL28469213

SCHEMBL28469213

O=Cc1cccn1Cc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.48
PPARA Q07869 2/20 0.48
ALDH1A1 P00352 3/20 0.46
TSHR P16473 1/20 0.44
CHRM5 P08912 1/20 0.42
GRM2 Q14416 2/20 0.42
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
KLKB1 P03952 1/20 0.40
TEAD1 P28347 1/20 0.40
MAPT P10636 1/20 0.40
SLC6A4 P31645 1/20 0.40
SERPINE1 P05121 2/20 0.39
PIM1 P11309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18002451 0.86 CHRM2 (0.47) EPHX2PPARAALDH1A1CHRM5GRM2
SCHEMBL18002488 0.83 ALDH1A1 (0.44) EPHX2PPARAALDH1A1MAPT
SCHEMBL1609235 0.80 ALDH1A1 (0.60) ALDH1A1MAPT
SCHEMBL17894535 0.80 ALDH1A1 (0.55) ALDH1A1CHRM5MAPT
SCHEMBL18002411 0.80 ALDH1A1 (0.41) ALDH1A1TSHRMAPT
SCHEMBL1609109 0.79 HDAC1 (0.56) EPHX2PPARAKLKB1TEAD1
SCHEMBL1609113 0.79 HDAC1 (0.56) EPHX2PPARAKLKB1TEAD1
SCHEMBL28469757 0.79 ALDH1A1 (0.54) ALDH1A1MAPT
SCHEMBL8136208 0.79 CYP11B1 (0.58) PPARAALDH1A1TSHRCHRM5TEAD1
SCHEMBL2056309 0.79 ALDH1A1 (0.50) EPHX2PPARAALDH1A1TSHRCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108358923-B Sophoridine pyrrole and indole derivatives, and preparation method and application thereof 广西大学 2020-11-03 CN claimed
CN-108047226-B Matrine pyrrole and indole derivatives, and preparation method and application thereof 广西大学 2020-11-03 CN claimed