SCHEMBL8136208

SCHEMBL8136208

O=Cc1cncn1Cc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.58
CYP11B2 P19099 6/20 0.58
FNTA P49354 3/20 0.43
PGGT1B P53609 3/20 0.43
FNTB P49356 2/20 0.43
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
CYP3A4 P08684 1/20 0.41
NAMPT P43490 1/20 0.40
CHRM5 P08912 2/20 0.40
TEAD1 P28347 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
HTR2C P28335 1/20 0.37
CPB1 P15086 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8134371 0.82 CYP11B1 (0.62) CYP11B1CYP11B2FNTAPGGT1BALDH1A1
SCHEMBL8129319 0.82 CYP11B2 (0.62) CYP11B1CYP11B2ALDH1A1
SCHEMBL8138765 0.81 CYP11B1 (0.58) CYP11B1CYP11B2ALDH1A1
SCHEMBL765399 0.80 CYP11B1 (0.67) CYP11B1CYP11B2ALDH1A1
SCHEMBL28469213 0.79 EPHX2 (0.48) ALDH1A1TSHRCHRM5TEAD1PPARA
SCHEMBL14476244 0.78 CYP11B1 (0.58) CYP11B1CYP11B2FNTAPGGT1B
SCHEMBL8131698 0.78 CYP11B1 (0.58) CYP11B1CYP11B2ALDH1A1
SCHEMBL1758083 0.78 CYP11B1 (0.68) CYP11B1CYP11B2ALDH1A1
SCHEMBL7660878 0.78 CYP11B1 (0.57) CYP11B1CYP11B2FNTAPGGT1BFNTB
SCHEMBL7986619 0.77 CYP11B1 (0.67) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054882-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 2000-11-29 EP disclosed
WO-1999041248-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AVENTIS PHARMA S.A. (FR) 1999-08-19 WO disclosed