SCHEMBL28470784

SCHEMBL28470784

Fc1ccc(-c2nc(-c3ccc4ccccc4n3)nc3ccccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.56
SCN9A Q15858 10/20 0.49
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
ATM Q13315 1/20 0.49
CYP19A1 P11511 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
AR P10275 1/20 0.43
KDM4E B2RXH2 2/20 0.42
GMNN O75496 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
THPO P40225 1/20 0.42
BLM P54132 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28924859 0.90 MEN1 (0.55) ADORA2AMEN1KMT2AATMNPC1
SCHEMBL28653132 0.86 ADORA2A (0.47) ADORA2ASCN9AMEN1KMT2AATM
SCHEMBL28466676 0.86 MEN1 (0.49) ADORA2AMEN1KMT2AATMAR
SCHEMBL28641606 0.86 MEN1 (0.49) MEN1KMT2AATMABCG2NPC1
SCHEMBL28633167 0.86 MEN1 (0.49) ADORA2AMEN1KMT2AATMABCG2
SCHEMBL28637623 0.85 MEN1 (0.46) ADORA2AMEN1KMT2AATMABCG2
SCHEMBL16436772 0.84 MEN1 (0.60) ADORA2AMEN1KMT2AATMNPC1
SCHEMBL28147443 0.82 MEN1 (0.71) ADORA2ASCN9AMEN1KMT2AATM
SCHEMBL28147464 0.82 MEN1 (0.71) ADORA2ASCN9AMEN1KMT2AATM
SCHEMBL8819242 0.81 TGFBR1 (0.55) ADORA2ASCN9AMEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110606839-B Green synthesis method of polysubstituted quinazoline derivative 南方医科大学 2021-10-08 CN claimed
CN-111700894-B Application of 2-azaarene substituted quinazoline compound in preparation of antitumor drugs 南方医科大学 2023-07-28 CN disclosed
CN-111700894-A Application of 2-azaarene substituted quinazoline compound in preparation of antitumor drugs 南方医科大学 2020-09-25 CN disclosed