SCHEMBL28477490

SCHEMBL28477490

O=[N+]([O-])c1cc(C(F)(F)F)[c]c(S(=O)(=O)N2CCNCC2)c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
ADRB1 P08588 1/20 0.36
SIRT6 Q8N6T7 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
IKBKB O14920 1/20 0.35
CHUK O15111 1/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSD11B1 P28845 1/20 0.34
USP2 O75604 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28482466 0.85 SMN1; SMN2 (0.44) SMN1; SMN2SIRT6LMNAALDH1A1HSD11B1
SCHEMBL28478897 0.83 ALDH1A1 (0.40) SMN1; SMN2PKMLMNAALDH1A1MEN1
SCHEMBL29202922 0.82 MAPT (0.52) MAPTLMNAALDH1A1KMT2A
SCHEMBL28482437 0.81 ALDH1A1 (0.43) SMN1; SMN2PKMLMNAALDH1A1KMT2A
SCHEMBL29202905 0.81 TRPV4 (0.40) SMN1; SMN2MAPTLMNAALDH1A1MEN1
SCHEMBL28473264 0.77 NPC1 (0.42) MAPTPKMLMNAALDH1A1MEN1
SCHEMBL1871493 0.68 MAPT (0.63) SMN1; SMN2ADRB1SIRT6MAPTPKM
Trifluoroacetic Acid SCHEMBL25303672 0.68 ALDH1A1 (0.54) SMN1; SMN2ADRB1SIRT6MAPTIKBKB
SCHEMBL28474493 0.67 HTT (0.47) SMN1; SMN2ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL28485486 0.67 HTT (0.47) SMN1; SMN2SIRT6MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111918864-A Prodrug compounds activated by AKR1C3 and their use to treat hyperproliferative disorders 阿基利斯医疗有限公司 2020-11-10 CN disclosed