SCHEMBL28477644

SCHEMBL28477644

NC(=O)OCCCCCNC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@@H]21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.68
PLCD1 P51178 1/20 0.62
CNR1 P21554 3/20 0.60
CA12 O43570 2/20 0.58
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA9 Q16790 2/20 0.58
F2 P00734 1/20 0.57
PRSS1 P07477 1/20 0.57
PRSS2 P07478 1/20 0.57
PRSS3 P35030 1/20 0.57
TPSAB1 Q15661 1/20 0.57
FOLH1 Q04609 2/20 0.56
CNR2 P34972 1/20 0.56
PKM P14618 2/20 0.56
MEN1 O00255 1/20 0.56
ABL1 P00519 1/20 0.56
LMNA P02545 1/20 0.56
IDE P14735 1/20 0.56
MAPK1 P28482 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8407567 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL31621058 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL13169001 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL19069314 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL18025829 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL24750115 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL5841368 0.90 TDP1 (0.76) TDP1PLCD1CA12CA1CA2
SCHEMBL18779801 0.89 TDP1 (0.78) TDP1PLCD1CA12CA1CA2
SCHEMBL8508187 0.89 TDP1 (0.71) TDP1PLCD1CNR1CA12CA1
SCHEMBL19960973 0.89 TDP1 (0.74) TDP1PLCD1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-A Diaryl substituted fused heterocyclic compound, preparation method thereof and application thereof in pharmacy 复旦大学 2020-10-02 CN disclosed