SCHEMBL28480271

SCHEMBL28480271

COC(=O)c1ccc(-n2c3ccc(-c4cnn(C5CCCCO5)c4)cc3c3cc(-c4cnn(C5CCCCO5)c4)ccc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.43
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
FGFR1 P11362 3/20 0.40
DDR2 Q16832 1/20 0.40
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
ALDH1A1 P00352 2/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FLT3 P36888 2/20 0.37
FGFR2 P21802 1/20 0.37
FGFR4 P22455 1/20 0.37
FGFR3 P22607 1/20 0.37
KDR P35968 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32662972 0.92 RXRA (0.44) MCL1RXRARXRBRXRGFGFR1
SCHEMBL28481979 0.89 MCL1 (0.46) MCL1RXRARXRBRXRGFGFR1
SCHEMBL23535723 0.87 MCL1 (0.45) MCL1RXRARXRBRXRGFGFR1
SCHEMBL29194155 0.81 RXRA (0.47) MCL1RXRARXRBRXRGFGFR1
SCHEMBL19029753 0.78 MCL1 (0.45) MCL1RXRARXRBRXRGFGFR1
SCHEMBL25167771 0.78 MCL1 (0.45) MCL1RXRARXRBRXRGFGFR1
SCHEMBL30867575 0.76 KDM5B (0.42) MCL1RXRARXRBRXRGFGFR1
SCHEMBL29194193 0.74 MCL1 (0.40) MCL1RXRARXRBRXRGFGFR1
SCHEMBL23535740 0.74 MCL1 (0.47) MCL1RXRARXRBRXRGFGFR1
SCHEMBL30041685 0.73 MKNK1 (0.46) MCL1RXRARXRBRXRGFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776504-B Metal organic framework material based on low-symmetry pyrazole-carboxylic acid ligand Zn, and preparation method and application thereof 北京工业大学 2020-10-16 CN claimed
CN-109776504-B Metal organic framework material based on low-symmetry pyrazole-carboxylic acid ligand Zn, and preparation method and application thereof 北京工业大学 2020-10-16 CN disclosed