SCHEMBL28480419

SCHEMBL28480419

O=C1CCc2ccc3c(ccc4ccccc43)c21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 4/20 0.50
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
HIF1A Q16665 2/20 0.49
MEN1 O00255 1/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP2D6 P10635 1/20 0.49
HPGD P15428 1/20 0.49
ALOX12 P18054 1/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 1/20 0.49
PAX8 Q06710 1/20 0.47
TDP1 Q9NUW8 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP2A6 P11509 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6759607 0.91 DNMT1 (0.44) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL30617063 0.91 DNMT1 (0.44) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL27619805 0.90 HPRT1 (0.47) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL17263921 0.82 PBRM1 (0.40) ALDH1A1MEN1USP2HPGDKMT2A
SCHEMBL6215591 0.80 ALDH1A1 (0.49) ALDH1A1MEN1USP2LMNAHPGD
SCHEMBL27467873 0.79 HPRT1 (0.47) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
Phthalazine SCHEMBL27577696 0.74 ALDH1A1 (0.49) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL29381793 0.74 HPRT1 (0.48) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL5672208 0.73 HPGD (0.44) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7345934 0.73 HPRT1 (0.58) HPRT1ALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111417410-A Glucocorticoid receptor agonists and immunoconjugates thereof 艾伯维公司 2020-07-14 CN disclosed