SCHEMBL28480511

SCHEMBL28480511

COC(=O)c1ccc(OCOCC[Si](C)(C)C)cc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.63
RAB9A P51151 4/20 0.56
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
SMN1; SMN2 Q16637 5/20 0.49
NPC1 O15118 3/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 3/20 0.46
GAA P10253 1/20 0.46
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
POLB P06746 2/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6041694 0.87 MAPT (0.48) MAPTRAB9ATDP1L3MBTL1SMN1; SMN2
SCHEMBL4912817 0.85 TDP1 (0.52) MAPTCA1CA2TDP1L3MBTL1
SCHEMBL6044419 0.85 CYSLTR1 (0.49) MAPTRAB9AL3MBTL1SMN1; SMN2NPC1
SCHEMBL3846345 0.84 L3MBTL1 (0.59) MAPTRAB9AL3MBTL1LMNAGAA
SCHEMBL5522952 0.84 PKM (0.53) RAB9AL3MBTL1SMN1; SMN2NPC1GAA
SCHEMBL4907075 0.84 MAPT (0.47) MAPTRAB9ATDP1L3MBTL1SMN1; SMN2
SCHEMBL28481517 0.84 CA1 (0.53) MAPTRAB9ACA1CA2SMN1; SMN2
SCHEMBL30427258 0.83 PARP10 (0.56) CA1CA2NPC1KMT2AALDH1A1
SCHEMBL1503528 0.83 MAPT (0.69) MAPTRAB9ACA1CA2TDP1
SCHEMBL11147412 0.81 MAPT (0.67) MAPTRAB9ACA1CA2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111875583-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-109666022-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-111875583-A Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2020-11-03 CN disclosed