SCHEMBL28484112

SCHEMBL28484112

c1c[nH]c(Nc2ccon2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
BACE1 P56817 1/20 0.33
GAPDH P04406 1/20 0.33
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3194321 0.72 DAO (0.35) GAA
SCHEMBL18796809 0.69
SCHEMBL5765529 0.68 KMT2A (0.50) SMN1; SMN2MEN1KMT2ATSHRGAA
SCHEMBL4792068 0.68 BRD4 (0.43) SMN1; SMN2GAA
SCHEMBL2012149 0.68 MEN1 (0.53) SMN1; SMN2MEN1KMT2AGAAHPGD
SCHEMBL19477810 0.67 MAPK10 (0.53) SMN1; SMN2MEN1KMT2AGAAPIK3CD
SCHEMBL10972199 0.67 GOT1 (0.47) PIK3CAMTOR
SCHEMBL28457161 0.67
SCHEMBL4667411 0.67 SCN9A (0.46) MEN1KMT2ABACE1RAB9AALDH1A1
SCHEMBL29463913 0.67 MAPK10 (0.53) SMN1; SMN2MEN1KMT2AGAAPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112074515-B Cyclic compounds as LPA antagonists isoxazoles of hexyl acid 百时美施贵宝公司 2025-01-10 CN disclosed
CN-112074515-A Cyclohexyl acid isoxazoles as LPA antagonists 百时美施贵宝公司 2020-12-11 CN disclosed