SCHEMBL28486193

SCHEMBL28486193

c1ccc(COc2n[nH]c3cncnc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.44
CNR2 P34972 3/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
MPO P05164 2/20 0.41
TPO P07202 1/20 0.41
CYP3A4 P08684 1/20 0.41
EPX P11678 1/20 0.41
MGMT P16455 1/20 0.41
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
MAPK1 P28482 3/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
SGMS2 Q8NHU3 1/20 0.39
FFAR2 O15552 1/20 0.38
DAPK1 P53355 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997227 0.76 TTK (0.50) CYP3A4CDC7MAPK1ALDH1A1HPGD
SCHEMBL28378989 0.76 PARP1 (0.43) MPOCYP3A4ALDH1A1HPGDHTT
SCHEMBL847077 0.70 LMNA (0.47) CNR1CNR2MGMTCDC7DBF4
SCHEMBL6997886 0.68 ALDH1A1 (0.46) CYP3A4MAPK1ALDH1A1LMNAHPGD
SCHEMBL5440113 0.68 KDM4C (0.47) MPOTPOCYP3A4EPXMGMT
SCHEMBL31261712 0.67 ALDH1A1 (0.48) CNR1CNR2CDC7DBF4MAPK1
SCHEMBL9980485 0.67 GRM4 (0.63) CYP3A4MAPK1TSHR
SCHEMBL22890209 0.67 CNR2 (0.52) CNR1CNR2HTR2CHTR2BMPO
SCHEMBL875608 0.67 LMNA (0.53) MAPK1LMNAL3MBTL1PRMT5
SCHEMBL1014840 0.66 CHEK1 (0.47) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010860-B Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2023-03-10 CN claimed
CN-112010860-A Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2020-12-01 CN claimed
CN-112010860-B Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2023-03-10 CN disclosed
CN-112010860-B Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2023-03-10 CN disclosed
CN-112010860-B Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2023-03-10 CN disclosed
CN-112010860-A Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2020-12-01 CN disclosed
CN-112010860-A Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2020-12-01 CN disclosed
CN-112010860-A Benzyloxypyrazolopyrimidine compounds, pharmaceutical compositions and uses thereof 南京纳丁菲医药科技有限公司 2020-12-01 CN disclosed