SCHEMBL2848652

SCHEMBL2848652

O=C(NCCc1cccc(F)c1)c1cnn(Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 9/20 0.56
SCD O00767 6/20 0.52
SCD5 Q86SK9 3/20 0.50
NAMPT P43490 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
LMNA P02545 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
TP53 P04637 1/20 0.49
GAA P10253 1/20 0.49
POLB P06746 1/20 0.48
THRB P10828 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2851988 0.88 KLKB1 (0.62) KLKB1SCD5NPC1RAB9A
SCHEMBL2857899 0.83 KLKB1 (0.56) KLKB1RAB9ALMNA
SCHEMBL2863128 0.82 TAAR1 (0.47) SCDSCD5NPC1RAB9ALMNA
SCHEMBL951879 0.80 POLB (0.60) KLKB1SCDSCD5TDP1POLB
SCHEMBL2850615 0.79 KLKB1 (0.73) KLKB1
SCHEMBL2854366 0.78 KLKB1 (0.80) KLKB1
SCHEMBL2857801 0.76 LMNA (0.67) KLKB1LMNA
SCHEMBL28614480 0.76 HIF1A (0.79) LMNAPOLBTHRB
SCHEMBL1972631 0.75 HDAC2 (0.71) NPC1RAB9ALMNATP53GAA
SCHEMBL16712957 0.73 ROCK1 (0.63) NAMPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed