SCHEMBL28492579

SCHEMBL28492579

COc1ccc(C(=O)n2cc(C=O)c3c(I)cccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
ACHE P22303 2/20 0.41
MGAM O43451 1/20 0.40
F12 P00748 1/20 0.40
AMY1A P0DUB6 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
CNR2 P34972 6/20 0.39
BCHE P06276 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KLK7 P49862 1/20 0.39
KLK14 Q9P0G3 1/20 0.39
KLK5 Q9Y337 1/20 0.39
HPGD P15428 1/20 0.38
BLM P54132 1/20 0.38
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
AKR1C3 P42330 2/20 0.36
AKR1C4 P17516 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28497701 0.86 PTGS2 (0.46) KMT2ABCHEALDH1A1HPGDPOLB
SCHEMBL28498848 0.86 KMT2A (0.48) KMT2AACHEMGAMF12AMY1A
SCHEMBL28505828 0.86 KMT2A (0.48) KMT2AACHEMGAMF12AMY1A
SCHEMBL28495147 0.85 PTGS2 (0.43) KMT2AACHEALDH1A1POLBL3MBTL1
SCHEMBL28495086 0.84 PTGS2 (0.46) KMT2AACHEF12POLBAKR1C3
SCHEMBL28496079 0.84 PTGS2 (0.46) KMT2AACHEMGAMAMY1AGAA
SCHEMBL28495418 0.83 PLAU (0.39) KMT2AALDH1A1HPGDPOLB
SCHEMBL28490523 0.83 HPGD (0.38) KMT2AALDH1A1HPGDPOLBL3MBTL1
SCHEMBL28490532 0.81 PTGS2 (0.48) KMT2AF12GAAALDH1A1HPGD
SCHEMBL28486883 0.80 KMT2A (0.69) KMT2AACHEALDH1A1BLMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112028811-A 4-iodo-indole compound and preparation method thereof 平顶山学院 2020-12-04 CN claimed
CN-112028811-B 4-iodo-indole compound and preparation method thereof 平顶山学院 2022-03-22 CN disclosed
CN-112028811-A 4-iodo-indole compound and preparation method thereof 平顶山学院 2020-12-04 CN disclosed