SCHEMBL2849368

SCHEMBL2849368

CCCc1nc(CC)c(-c2ccc(OC(F)(F)F)cc2)c(=O)n1Cc1ccc(-c2ccccc2)c(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.44
CYP19A1 P11511 1/20 0.40
CHRM5 P08912 1/20 0.40
AGTR1 P30556 3/20 0.39
AGTR2 P50052 2/20 0.39
XDH P47989 1/20 0.39
PDE8A O60658 1/20 0.37
PDE7A Q13946 1/20 0.37
PDE7B Q9NP56 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1887930 0.91 PPARG (0.54) PPARGAGTR1AGTR2
SCHEMBL12357098 0.82 PPARG (0.53) PPARGAGTR1AGTR2
SCHEMBL4012974 0.81 PPARG (0.48) PPARGCYP19A1AGTR1AGTR2
SCHEMBL1892312 0.81 PPARG (0.58) PPARGAGTR1
SCHEMBL1890655 0.79 PPARG (0.56) PPARGAGTR1AGTR2
SCHEMBL1891285 0.79 PPARG (0.54) PPARGAGTR1
SCHEMBL4164574 0.79 PPARG (0.60) PPARGAGTR1AGTR2
SCHEMBL4010303 0.79 PPARG (0.55) PPARGAGTR1AGTR2
SCHEMBL1889130 0.78 PPARG (0.49) PPARGAGTR1
SCHEMBL12349090 0.77 AGTR1 (0.46) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2256115-A1 Heteromonocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-12-01 EP disclosed