SCHEMBL28495362

SCHEMBL28495362

Fc1cc2c(Cl)cc(Cl)nc2cc1Br

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.37
KDM1A O60341 2/20 0.34
KDM1B Q8NB78 2/20 0.34
MAPT P10636 1/20 0.33
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636878 0.82 NT5E (0.36) NT5EMAPTLMNA
SCHEMBL30656089 0.82 NT5E (0.36) NT5EMAPTLMNA
SCHEMBL20641687 0.82 KDM1A (0.36) NT5EKDM1AKDM1BMAPTESR1
SCHEMBL29487315 0.74 HTT (0.35) KDM1AKDM1B
SCHEMBL2724749 0.74 HTT (0.35) KDM1AKDM1B
SCHEMBL14690825 0.74 MAPT (0.40) NT5EMAPTESR1ESR2LMNA
SCHEMBL28499601 0.74 AXL (0.38) MAPT
SCHEMBL15647874 0.74 EGFR (0.38) MAPT
SCHEMBL26998825 0.73 ACHE (0.40) NT5EMAPTESR1ESR2LMNA
SCHEMBL24252971 0.73 KDM1A (0.33) KDM1AKDM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112110918-B Spiro substituted pyrimido cyclic compounds, process for their preparation and their use in medicine 劲方医药科技(上海)有限公司 2023-08-22 CN disclosed
CN-112110918-A Spiro-substituted pyrimido-cyclic compounds, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2020-12-22 CN disclosed