SCHEMBL28500191

SCHEMBL28500191

CC(=O)c1c(C)c2ccc(OS(=O)(=O)C(F)(F)F)cc2oc1=O

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.61
HPGD P15428 2/20 0.54
STS P08842 1/20 0.53
MAOB P27338 2/20 0.52
ALPL P05186 6/20 0.50
ALPI P09923 5/20 0.50
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
RAB9A P51151 1/20 0.48
MAOA P21397 1/20 0.47
ALDH1A2 O94788 1/20 0.47
ALDH1B1 P30837 1/20 0.47
ALDH1A3 P47895 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10847170 0.86 HPGD (0.72) HSD11B1HPGDSTSMAOBALPL
SCHEMBL28510448 0.81 HSD11B1 (0.53) HSD11B1STSRAB9A
SCHEMBL30507295 0.81 HSD11B1 (0.53) HSD11B1STSRAB9A
SCHEMBL28508245 0.80 HSD11B1 (0.52) HSD11B1
SCHEMBL28508234 0.80 HSD11B1 (0.52) HSD11B1
SCHEMBL28500203 0.80 HSD11B1 (0.52) HSD11B1HPGDSTSMAOB
SCHEMBL30507233 0.80 HSD11B1 (0.52) HSD11B1
SCHEMBL18493227 0.79 KDM4E (0.68) HPGDSTSALDH1A1KDM4ECYP2C9
SCHEMBL2772042 0.78 HSD11B1 (0.50) HSD11B1HPGDSTSMAOBALDH1A1
SCHEMBL13155387 0.77 HSD11B1 (0.48) HSD11B1HPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-B Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2023-07-25 CN disclosed
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed