SCHEMBL28501669

SCHEMBL28501669

CNc1cccc(-c2ccnc(N)n2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.58
HSP90AA1 P07900 2/20 0.57
AURKA O14965 2/20 0.57
PRKACA P17612 2/20 0.57
ADORA2A P29274 1/20 0.57
HSP90AB1 P08238 1/20 0.51
PTK2 Q05397 1/20 0.51
KMO O15229 1/20 0.50
CDK2 P24941 3/20 0.45
CCNT1 O60563 2/20 0.45
CCNA2 P20248 2/20 0.45
CDK9 P50750 2/20 0.45
CAMK2D Q13557 1/20 0.45
LARS1 Q9P2J5 1/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 2/20 0.44
CHUK O15111 1/20 0.44
PDPK1 O15530 1/20 0.44
RPS6KB1 P23443 1/20 0.44
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312358 0.83 PLK1 (0.59) PLK1KMOCDK9KDRALDH1A1
SCHEMBL4708076 0.78 HSP90AA1 (0.67) PLK1HSP90AA1AURKAPRKACAADORA2A
SCHEMBL16285520 0.78 PLK1 (0.52) PLK1NPC1RAB9AMEN1KMT2A
SCHEMBL4202167 0.77 HSP90AA1 (0.76) HSP90AA1AURKAPRKACAADORA2AHSP90AB1
SCHEMBL5229810 0.76 HSP90AA1 (0.62) HSP90AA1AURKAPRKACAADORA2AHSP90AB1
SCHEMBL6764764 0.76 HSP90AA1 (0.62) PLK1HSP90AA1AURKAPRKACAADORA2A
SCHEMBL481304 0.76 PRKACA (0.62) HSP90AA1AURKAPRKACAADORA2AHSP90AB1
SCHEMBL15650217 0.75 ADORA2A (0.57) HSP90AA1AURKAPRKACAADORA2AHSP90AB1
SCHEMBL16285497 0.75 PLK1 (0.50) PLK1KDRSYKALDH1A1MAPT
SCHEMBL316210 0.74 HSP90AA1 (1.00) HSP90AA1AURKAPRKACAADORA2AHSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed