SCHEMBL4202167

SCHEMBL4202167

Nc1nccc(-c2cccc(-c3ccccc3)c2)n1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.76
ADORA2A P29274 2/20 0.76
AURKA O14965 2/20 0.76
PRKACA P17612 1/20 0.76
HSP90AB1 P08238 1/20 0.57
PTK2 Q05397 1/20 0.57
KMO O15229 1/20 0.56
ROCK1 Q13464 2/20 0.53
MAPK13 O15264 1/20 0.51
RAF1 P04049 1/20 0.51
MAPK9 P45984 1/20 0.51
MAPK12 P53778 1/20 0.51
MAPK11 Q15759 1/20 0.51
MAPK14 Q16539 1/20 0.51
ADORA1 P30542 1/20 0.50
CDK2 P24941 4/20 0.49
HRH4 Q9H3N8 1/20 0.49
CHUK O15111 1/20 0.49
PDPK1 O15530 1/20 0.49
RPS6KB1 P23443 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12176972 0.87 HSP90AA1 (0.92) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
SCHEMBL316210 0.87 HSP90AA1 (1.00) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
Hydrochloric Acid SCHEMBL17186384 0.85 HSP90AA1 (0.96) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
SCHEMBL4708076 0.84 HSP90AA1 (0.67) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
SCHEMBL13977116 0.83 HSP90AA1 (0.57) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
SCHEMBL1448939 0.82 HSP90AA1 (0.65) HSP90AA1ADORA2AAURKAPRKACAHSP90AB1
SCHEMBL19781417 0.81 MEN1 (0.54) HSP90AA1ADORA2AAURKAPRKACAKMO
SCHEMBL18134284 0.81 KMT2A (0.58) HSP90AA1ADORA2AAURKAPRKACAKMO
SCHEMBL18731939 0.81 KMT2A (0.58) HSP90AA1ADORA2AAURKAPRKACAKMO
SCHEMBL18134295 0.81 KMT2A (0.58) HSP90AA1ADORA2AAURKAPRKACAKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011136483-A1 NOVEL COMPOUNDS FOR ORGANIC ELECTRONIC MATERIAL AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2011-11-03 WO disclosed
EP-2032543-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES Boehringer Ingelheim International GmbH (DE) 2009-03-11 EP disclosed
WO-2007146977-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed