SCHEMBL28501937

SCHEMBL28501937

CC#CNC(=O)c1cn(-c2ccccc2)nc1-c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 3/20 0.65
AURKA O14965 9/20 0.64
TP53 P04637 1/20 0.64
MAPT P10636 3/20 0.62
LMNA P02545 3/20 0.61
GAA P10253 1/20 0.61
KMT2A Q03164 3/20 0.58
MEN1 O00255 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
ALDH1A1 P00352 3/20 0.58
KDM4E B2RXH2 1/20 0.58
PLA2G1B P04054 1/20 0.55
ATG4B Q9Y4P1 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
CDK2 P24941 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6256569 0.82 AURKA (0.72) KDM5BAURKATP53MAPTLMNA
SCHEMBL976547 0.81 AURKA (0.74) KDM5BAURKATP53MAPTLMNA
SCHEMBL22095269 0.79 AURKA (1.00) KDM5BAURKATP53MAPTLMNA
SCHEMBL4501557 0.77 ALDH1A1 (0.82) KDM5BAURKATP53MAPTLMNA
SCHEMBL12264890 0.77 MAPT (1.00) KDM5BAURKATP53MAPTLMNA
SCHEMBL14132504 0.76 TP53 (0.73) KDM5BAURKATP53MAPTLMNA
SCHEMBL22095286 0.76 KDM5B (0.95) KDM5BAURKATP53MAPTLMNA
SCHEMBL14132445 0.75 KDM5B (0.69) KDM5BAURKATP53MAPTLMNA
SCHEMBL28771391 0.75 ALDH1A1 (0.78) KDM5BAURKATP53MAPTLMNA
SCHEMBL5812722 0.75 MAPT (0.67) KDM5BAURKATP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109970654-B A series of substituted 2-phenyl pyrazole derivatives, and preparation method and application thereof 郑州大学 2020-12-25 CN disclosed