SCHEMBL6256569

SCHEMBL6256569

CNC(=O)c1cn(-c2ccccc2)nc1-c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AURKA O14965 9/20 0.72
TP53 P04637 1/20 0.72
MAPT P10636 3/20 0.70
KDM5B Q9UGL1 3/20 0.68
LMNA P02545 3/20 0.68
GAA P10253 1/20 0.68
KMT2A Q03164 3/20 0.64
MEN1 O00255 2/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
ALDH1A1 P00352 4/20 0.64
KDM4E B2RXH2 1/20 0.64
PLA2G1B P04054 1/20 0.60
ATG4B Q9Y4P1 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL976547 0.87 AURKA (0.74) AURKATP53MAPTKDM5BLMNA
SCHEMBL23928535 0.86 AURKA (0.78) AURKATP53MAPTLMNAGAA
SCHEMBL22095269 0.84 AURKA (1.00) AURKATP53MAPTKDM5BLMNA
SCHEMBL4501557 0.83 ALDH1A1 (0.82) AURKATP53MAPTKDM5BLMNA
SCHEMBL28501937 0.82 KDM5B (0.65) AURKATP53MAPTKDM5BLMNA
SCHEMBL12264890 0.82 MAPT (1.00) AURKATP53MAPTKDM5BLMNA
SCHEMBL14132504 0.82 TP53 (0.73) AURKATP53MAPTKDM5BLMNA
SCHEMBL22095286 0.81 KDM5B (0.95) AURKATP53MAPTKDM5BLMNA
SCHEMBL14132445 0.80 KDM5B (0.69) AURKATP53MAPTKDM5BLMNA
SCHEMBL5812722 0.80 MAPT (0.67) AURKATP53MAPTKDM5BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005061462-A2 DIARYL PYRAZOLE DERIVATIVES AND THEIR USE AS NEUROKININ-3 RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2005-07-07 WO disclosed