SCHEMBL2850207

SCHEMBL2850207

O=C(O)NCCc1cccc(NC(=O)NCCCc2ccccc2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.72
KDM4E B2RXH2 1/20 0.72
KMT2A Q03164 7/20 0.70
MEN1 O00255 4/20 0.70
SMN1; SMN2 Q16637 4/20 0.70
ALDH1A1 P00352 3/20 0.70
LMNA P02545 3/20 0.70
HTT P42858 2/20 0.70
TP53 P04637 1/20 0.70
NPC1 O15118 4/20 0.66
RAB9A P51151 4/20 0.66
MAPT P10636 2/20 0.66
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C9 P11712 2/20 0.64
CYP2C19 P33261 2/20 0.64
CA12 O43570 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CA9 Q16790 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826334 0.96 KMT2A (0.75) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL2827311 0.95 KMT2A (0.72) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL2849248 0.88 MEN1 (0.62) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL1206194 0.87 KDM4E (0.72) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL2824601 0.86 NPC1 (0.61) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL12196188 0.84 EPHX1 (1.00) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL1204443 0.84 KMT2A (0.69) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL1205663 0.83 KMT2A (0.71) EPHX1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL8059186 0.83 KMT2A (0.55) KMT2AMEN1SMN1; SMN2ALDH1A1LMNA
SCHEMBL10192070 0.82 KMT2A (0.82) EPHX1KDM4EKMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed