SCHEMBL28503221

SCHEMBL28503221

CC(C)(C)OC(=O)N(C(=O)O)C(C)(C)Cc1ccc(C(F)(F)F)c(Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 8/20 0.40
CACNA1B Q00975 2/20 0.35
CACNA1C Q13936 2/20 0.35
CACNA1G O43497 1/20 0.35
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
HTT P42858 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
CACNA1H O95180 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29242138 0.81 XPO1 (0.47) XPO1CNR2
SCHEMBL855385 0.76 XPO1 (0.43) XPO1CACNA1BCACNA1CCACNA1GHTT
SCHEMBL27627602 0.75 XPO1 (0.42) XPO1HTT
SCHEMBL22028970 0.75 XPO1 (0.49) XPO1CACNA1BCACNA1CCACNA1GHTT
SCHEMBL29028016 0.74 SSTR4 (0.34)
SCHEMBL28379002 0.74 AKT1 (0.36) HTR2CSLC6A4HDAC1CNR2
SCHEMBL22029019 0.74 XPO1 (0.48) XPO1CACNA1BCACNA1CCACNA1GHTT
SCHEMBL30911244 0.74 XPO1 (0.48) XPO1CACNA1BCACNA1CCACNA1GHTT
SCHEMBL28512757 0.72 XPO1 (0.45) XPO1HTT
SCHEMBL28176575 0.68 AKT1 (0.41) XPO1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112105419-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-29 CN disclosed
CN-112105419-A Fused ring compound 豪夫迈·罗氏有限公司 2020-12-18 CN disclosed