SCHEMBL28504133

SCHEMBL28504133

COC(=O)C(N)CCc1nnnn1CCC#N

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NAALAD2 Q9Y3Q0 3/20 0.60
GHSR Q92847 3/20 0.38
TDP1 Q9NUW8 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21515089 1.00 NAALAD2 (0.60) NAALAD2GHSRTDP1TRPV1
Hydrochloric Acid SCHEMBL28501489 0.99 NAALAD2 (0.58) NAALAD2GHSRTDP1
Hydrochloric Acid SCHEMBL21494731 0.99 NAALAD2 (0.58) NAALAD2GHSRTDP1
SCHEMBL23030236 0.88 NAALAD2 (0.46) NAALAD2TRPV1
Chloromethane SCHEMBL29231841 0.84 NAALAD2 (0.64) NAALAD2GHSR
Hydrochloric Acid SCHEMBL21494705 0.84 NAALAD2 (0.67) NAALAD2GHSR
Hydrochloric Acid SCHEMBL21494707 0.84 NAALAD2 (0.67) NAALAD2GHSR
SCHEMBL14102932 0.82 NAALAD2 (0.53) NAALAD2GHSR
SCHEMBL21515088 0.79 NAALAD2 (0.60) NAALAD2GHSR
SCHEMBL28513600 0.79 NAALAD2 (0.60) NAALAD2GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218858-A 2, 6-diamino-3, 4-dihydropyrimidin-4-one derivatives and their use in therapy 托马斯·黑勒戴药物研究基金会 2021-01-12 CN disclosed