SCHEMBL28504451

SCHEMBL28504451

COc1cc(B2OC(C)(C)C(C)(C)O2)cc(OC)c1N1CCN(C2CCN(C)CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
HTR1A P08908 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
ACVR1 Q04771 1/20 0.34
FGFR3 P22607 1/20 0.34
KCNH2 Q12809 1/20 0.34
KDM4E B2RXH2 6/20 0.33
HTT P42858 1/20 0.33
EHMT2 Q96KQ7 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TRPV6 Q9H1D0 1/20 0.32
CCR4 P51679 1/20 0.32
DCLK1 O15075 1/20 0.32
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28514928 0.88 CCR4 (0.39) SMN1; SMN2CCR4
SCHEMBL28509497 0.84 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2
SCHEMBL28502237 0.83 ALDH1A1 (0.37) ALDH1A1
SCHEMBL26702882 0.81 FGFR3 (0.45) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL28504440 0.81 CCR4 (0.39) ALDH1A1KDM4EHTTCCR4
SCHEMBL28502430 0.80 CCR4 (0.36) ALDH1A1HTR1AKDM4ECCR4
SCHEMBL28503601 0.77 ALDH1A1 (0.41) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL15375421 0.77 ALDH1A1 (0.44) ALDH1A1KDM4E
SCHEMBL16826628 0.74 ALDH1A1 (0.40) ALDH1A1ACVR1TRPV6
SCHEMBL19099105 0.73 MEN1 (0.38) ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed